Research use only.  Educational reference. Not medical advice. Not for human consumption.
📈 Selective GH Secretagogue

Ipamorelin (10 mg Vial) Dosage Protocol

Ipamorelin is a selective GHRP (growth hormone releasing peptide) that stimulates GH secretion without significant cortisol or prolactin elevation — the cleanest of the GHRP class.

⚡ Quickstart Highlights

Vial size
10 mg
Reconstitution
3 mL BAC water → 3.33 mg/mL
1 U-100 unit =
33.3 mcg
Frequency
1–3× daily

Dosing & Reconstitution Guide

Route: Subcutaneous  |  Frequency: 1–3× daily  |  Half-life: ~2 hours

Standard Approach (3 mL = 3.33 mg/mL)

Reconstituting with 3 mL bacteriostatic water produces a concentration of 3.33 mg/mL. Volume per dose changes with concentration; mg dose itself does not change between vial sizes.

Phase / ProtocolDoseU-100 UnitsVolumeDoses per vial
Weeks 1–2 (titration)100 mcg3 units0.030 mL100 doses
Weeks 3–4150 mcg4.5 units0.045 mL66 doses
Weeks 5–8200 mcg6 units0.060 mL50 doses
Weeks 9–12 (maintenance)250 mcg7.5 units0.075 mL40 doses

Reconstitution Steps

  1. Wipe the vial stopper and BAC water vial with alcohol; let dry.
  2. Draw 3 mL of bacteriostatic water into a sterile syringe.
  3. Inject slowly down the inside glass wall of the peptide vial. Do not aim at the powder.
  4. Gently swirl until fully dissolved. Do not shake.
  5. Label with reconstitution date. Refrigerate at 2–8°C; use within 28 days.

Supplies Needed

Estimates for an 8-week and 12-week cycle at 250 mcg per dose, 1–3× daily (3 doses/week).

Item8-Week Cycle12-Week Cycle
Ipamorelin (10 mg) vials1 vials1 vials
Insulin syringes (U-100)2436
Bacteriostatic water (10 mL)1 × 10 mL1 × 10 mL
Alcohol swabs1 × 100-pack2 × 100-pack

Protocol Overview

Ipamorelin is the cleanest GHRP — meaning it stimulates GH release without significant cortisol or prolactin elevation. This makes it the GHRP of choice for sustained-use protocols where cortisol elevation would be unwanted (recovery, sleep, anti-aging).

Almost always paired with a GHRH analog (CJC-1295 no-DAC, sermorelin, or tesamorelin) for the synergistic pulse amplification effect. Solo ipamorelin produces a measurable but modest GH pulse.

Dosing Protocol

Dosing by intensity:

Cycle structure: 12–16 weeks continuous, 4-week break. Receptor desensitization is uncommon at clean ipamorelin doses but cycling is the conservative default.

Stacking: Almost always combined with a GHRH analog. See CJC-1295 + Ipamorelin or Tesamorelin + Ipamorelin blends.

Timing: Avoid eating for 30+ min after dose. Pre-bed timing aligns with natural overnight GH pulse.

Storage Instructions

StateTemperatureDuration
Lyophilized−20°C (−4°F)Up to 24 months, dry & dark
Reconstituted2–8°C (35–46°F)Up to 28 days, protect from light

Important Notes

⚠ Research Use Only: Ipamorelin is investigational.

How This Works

Ipamorelin is a 5-amino-acid synthetic peptide that mimics ghrelin at the growth-hormone secretagogue receptor (GHS-R1a) on pituitary somatotrophs. Activation triggers release of stored GH.

Unlike GHRP-2 and GHRP-6, ipamorelin shows minimal effect on cortisol, prolactin, or ACTH at therapeutic doses — making it the "cleanest" of the GHRP class. It pairs synergistically with GHRH analogs (CJC-1295, sermorelin) which stimulate via the GHRH receptor.

Potential Benefits & Side Effects

Potential Benefits

Side Effect Profile

Lifestyle Factors

Injection Technique

References

1
Raun K et al. 'Ipamorelin: a potent and selective growth hormone secretagogue' — Eur J Endocrinol, 1998 View source ↗